SCHEMBL5369563

SCHEMBL5369563

C[Si](C)(C)CCOCn1c(C(=O)O)nc2cccc(CBr)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ELANE P08246 9/20 0.42
NPC1 O15118 1/20 0.38
F11 P03951 1/20 0.32
PIK3CD O00329 1/20 0.31
KLKB1 P03952 1/20 0.31
MAPT P10636 1/20 0.30
AKR1B10 O60218 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4932747 0.88 ELANE (0.43) ELANENPC1
SCHEMBL7823682 0.85 ELANE (0.45) ELANENPC1
SCHEMBL5381357 0.84 NPC1 (0.35) NPC1KLKB1
SCHEMBL17324961 0.81 ELANE (0.43) ELANEMAPT
SCHEMBL5374515 0.80 NPC1 (0.37) ELANENPC1F11KLKB1MAPT
SCHEMBL4935725 0.77 MMP13 (0.40) NPC1MAPT
SCHEMBL4935109 0.75 CASR (0.39) ELANENPC1
SCHEMBL4934889 0.73 SMN1; SMN2 (0.38) NPC1MAPT
SCHEMBL1314051 0.71 NPC1 (0.35) NPC1F11KLKB1MAPT
SCHEMBL7815551 0.71 HRH3 (0.43) ELANENPC1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed