SCHEMBL5374982

SCHEMBL5374982

O=c1ccc(Cc2cc(Oc3cccc(Cl)c3)c3occc3c2)n[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 1.00
RHEB Q15382 2/20 0.34
SLC6A4 P31645 3/20 0.33
AKR1B1 P15121 1/20 0.33
HTR2A P28223 1/20 0.33
KCNH2 Q12809 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
AHR P35869 1/20 0.32
PDE4B Q07343 2/20 0.32
MAPK8 P45983 1/20 0.32
PDE5A O76074 1/20 0.32
PDE9A O76083 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5372498 0.91 CYP3A4 (0.83) CYP3A4AKR1B1THRATHRB
SCHEMBL5377164 0.89 CYP3A4 (0.80) CYP3A4RHEBSLC6A4AKR1B1HTR2A
SCHEMBL5370307 0.89 CYP3A4 (0.80) CYP3A4AKR1B1THRATHRB
SCHEMBL5368948 0.86 CYP3A4 (0.75) CYP3A4PRMT5WDR77
SCHEMBL5372604 0.83 CYP3A4 (0.71) CYP3A4THRATHRBADORA3ADORA2A
SCHEMBL5371235 0.83 CYP3A4 (0.71) CYP3A4THRATHRB
SCHEMBL5375849 0.80 CYP3A4 (0.67) CYP3A4
SCHEMBL5365181 0.80 CYP3A4 (0.67) CYP3A4RHEBSLC6A4AKR1B1HTR2A
SCHEMBL5367092 0.80 CYP3A4 (0.66) CYP3A4RHEBSLC6A4AKR1B1HTR2A
SCHEMBL5377723 0.79 CYP3A4 (0.66) CYP3A4RHEBSLC6A4AKR1B1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed