SCHEMBL5368948

SCHEMBL5368948

N#Cc1cccc(Oc2cc(Cc3ccc(=O)[nH]n3)cc3ccoc23)c1

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.75
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
CYP11B1 P15538 12/20 0.34
CYP11B2 P19099 8/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
P2RX3 P56373 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5375849 0.90 CYP3A4 (0.67) CYP3A4CYP11B1CYP11B2MAOAMAOB
SCHEMBL5370307 0.86 CYP3A4 (0.80) CYP3A4
SCHEMBL5374982 0.86 CYP3A4 (1.00) CYP3A4PRMT5WDR77
SCHEMBL5372498 0.81 CYP3A4 (0.83) CYP3A4
SCHEMBL5377164 0.81 CYP3A4 (0.80) CYP3A4CYP11B1CYP11B2MAOAMAOB
SCHEMBL5372604 0.81 CYP3A4 (0.71) CYP3A4MAOA
SCHEMBL5371235 0.81 CYP3A4 (0.71) CYP3A4
SCHEMBL5377579 0.80 CYP3A4 (0.52) CYP3A4FNTAFNTBPGGT1BPRMT5
SCHEMBL5374410 0.80 CYP3A4 (0.49) CYP3A4FNTAFNTBPGGT1BPRMT5
SCHEMBL5370328 0.80 CYP3A4 (0.47) CYP3A4FNTAFNTBPGGT1BPRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed