SCHEMBL5372604

SCHEMBL5372604

Cc1cc(C)cc(Oc2cc(Cc3ccc(=O)[nH]n3)cc3ccoc23)c1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.71
MAOA P21397 1/20 0.32
THRA P10827 2/20 0.32
THRB P10828 2/20 0.32
MAPT P10636 1/20 0.32
LMNA P02545 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371235 0.88 CYP3A4 (0.71) CYP3A4THRATHRB
SCHEMBL5372498 0.88 CYP3A4 (0.83) CYP3A4THRATHRBKDM4ENPC1
SCHEMBL5370307 0.87 CYP3A4 (0.80) CYP3A4THRATHRB
SCHEMBL5377164 0.85 CYP3A4 (0.80) CYP3A4MAOATHRATHRBKDM4E
SCHEMBL5374982 0.83 CYP3A4 (1.00) CYP3A4THRATHRBADORA3ADORA2A
SCHEMBL5375849 0.83 CYP3A4 (0.67) CYP3A4MAOA
SCHEMBL5385611 0.81 CYP3A4 (0.62) CYP3A4
SCHEMBL5368948 0.81 CYP3A4 (0.75) CYP3A4MAOA
SCHEMBL5376979 0.80 CYP3A4 (0.61) CYP3A4MAOAMAPTLMNA
SCHEMBL5373845 0.75 CYP3A4 (0.40) CYP3A4THRATHRBLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed