SCHEMBL5375034

SCHEMBL5375034

N#Cc1ccc(C(F)(F)F)c(Oc2cc(Cc3ccc(=O)[nH]n3)ccc2Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.37
KDR P35968 2/20 0.35
TRPV4 Q9HBA0 1/20 0.34
KCNH2 Q12809 2/20 0.34
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ESRRB O95718 1/20 0.33
ESR1 P03372 1/20 0.33
ESRRA P11474 1/20 0.33
ESRRG P62508 1/20 0.33
ESR2 Q92731 1/20 0.33
AR P10275 1/20 0.33
SLC22A12 Q96S37 3/20 0.33
S100A9 P06702 1/20 0.32
CETP P11597 1/20 0.32
HTR2A P28223 1/20 0.32
MRGPRX4 Q96LA9 2/20 0.31
NTRK1 P04629 1/20 0.31
CYP19A1 P11511 1/20 0.31
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370850 0.91 CYP3A4 (0.42) CYP3A4TRPV4KCNH2CYP2C9CYP2C19
SCHEMBL5373721 0.86 CYP3A4 (0.39) CYP3A4KCNH2CYP2C9CYP2C19SLC22A12
SCHEMBL5377021 0.86 AR (0.41) CYP3A4KCNH2CYP2C9CYP2C19ESRRA
SCHEMBL14559753 0.85 AR (0.39) CYP3A4TRPV4KCNH2CYP2C9CYP2C19
SCHEMBL5374211 0.85 CYP3A4 (0.38) CYP3A4KCNH2CYP2C9CYP2C19ESRRA
SCHEMBL5365226 0.84 SLC22A12 (0.40) CYP3A4KCNH2CYP2C9CYP2C19ESRRA
SCHEMBL5374946 0.84 CYP3A4 (0.42) CYP3A4KDRARNTRK1DAO
SCHEMBL5373732 0.84 CYP3A4 (0.45) CYP3A4KCNH2CYP2C9CYP2C19AR
SCHEMBL5375891 0.83 CYP3A4 (0.38) CYP3A4KCNH2CYP2C9CYP2C19ESRRA
SCHEMBL5366785 0.83 AR (0.41) CYP3A4KCNH2CYP2C9CYP2C19ESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed