SCHEMBL5373732

SCHEMBL5373732

N#Cc1cccc(Oc2cc(Cc3ccc(=O)[nH]n3)ccc2C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.45
EPAS1 Q99814 3/20 0.38
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PGGT1B P53609 1/20 0.38
VEGFA P15692 1/20 0.38
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
AR P10275 6/20 0.36
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SCN9A Q15858 4/20 0.34
KCNH2 Q12809 1/20 0.34
MEN1 O00255 1/20 0.34
CNR1 P21554 1/20 0.34
GPR183 P32249 1/20 0.34
CNR2 P34972 1/20 0.34
KMT2A Q03164 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374410 0.87 CYP3A4 (0.49) CYP3A4EPAS1FNTAFNTBPGGT1B
SCHEMBL5366909 0.86 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19
SCHEMBL5374482 0.85 CYP3A4 (0.61) CYP3A4EPAS1FNTAFNTBPGGT1B
SCHEMBL5377579 0.85 CYP3A4 (0.52) CYP3A4EPAS1FNTAFNTBPGGT1B
SCHEMBL5375295 0.85 CYP3A4 (0.47) CYP3A4EPAS1FNTAFNTBPGGT1B
SCHEMBL5370328 0.85 CYP3A4 (0.47) CYP3A4EPAS1FNTAFNTBPGGT1B
SCHEMBL5370543 0.84 CYP3A4 (0.46) CYP3A4EPAS1FNTAFNTBPGGT1B
SCHEMBL5375034 0.84 CYP3A4 (0.37) CYP3A4ARCYP2C9CYP2C19KCNH2
SCHEMBL5368699 0.82 AR (0.39) CYP3A4PRMT5WDR77AR
SCHEMBL5377568 0.80 CYP3A4 (0.47) CYP3A4ARCYP2C9CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed