SCHEMBL5375202

SCHEMBL5375202

O=C(O)c1cc(S(=O)(=O)Nc2ccc(OCc3ccccc3)cc2)ccc1O

nearest known ligand 0.78

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.78
KMT2A Q03164 5/20 0.78
PKM P14618 1/20 0.78
AR P10275 8/20 0.65
POLB P06746 2/20 0.62
TDP1 Q9NUW8 1/20 0.62
PGR P06401 1/20 0.61
MCL1 Q07820 1/20 0.61
ALDH1A1 P00352 3/20 0.61
GPR55 Q9Y2T6 1/20 0.56
KDM4E B2RXH2 1/20 0.56
TSHR P16473 1/20 0.55
ACLY P53396 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19329686 0.91 MEN1 (0.69) MEN1KMT2APKMARPOLB
SCHEMBL5371903 0.88 MEN1 (0.77) MEN1KMT2APKMARPOLB
SCHEMBL5380382 0.88 MEN1 (0.77) MEN1KMT2APKMARPOLB
SCHEMBL5373189 0.86 MEN1 (0.77) MEN1KMT2APKMARPOLB
SCHEMBL5378751 0.85 MEN1 (0.72) MEN1KMT2APKMARPOLB
SCHEMBL11222668 0.83 ALDH1A1 (0.75) MEN1KMT2APKMPOLBMCL1
SCHEMBL665516 0.82 AR (0.78) MEN1KMT2APKMARPOLB
SCHEMBL5368222 0.81 MEN1 (1.00) MEN1KMT2APKMARPOLB
SCHEMBL3504223 0.81 ALDH1A1 (0.65) MEN1KMT2APOLBALDH1A1KDM4E
SCHEMBL1249879 0.81 POLB (0.77) MEN1KMT2APOLBMCL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7262318-B2 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER, INC. (US) 2007-08-28 US disclosed
US-7262318-B2 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER, INC. (US) 2007-08-28 US disclosed
US-7262318-B2 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER, INC. (US) 2007-08-28 US disclosed
US-20060258723-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds PFIZER INC 2006-11-16 US disclosed
US-20050228015-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER INC 2005-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050228015-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PPARA, PPARG, PPARD MEN1 4855/4885KMT2A 3530/4885PKM 861/4885
US-20060258723-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds PPARG, PPARA, PPARD MEN1 4861/4885KMT2A 3601/4885PKM 859/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.