SCHEMBL5375238

SCHEMBL5375238

COc1cc(-c2cc(=O)[nH]c(-c3ccncc3)n2)ccn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 6/20 0.60
IDO1 P14902 1/20 0.49
MAPT P10636 1/20 0.48
AKT1 P31749 1/20 0.46
CYP19A1 P11511 1/20 0.45
DYRK1A Q13627 1/20 0.44
PKN1 Q16512 1/20 0.44
PKN2 Q16513 1/20 0.44
POLB P06746 1/20 0.42
CDC7 O00311 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
PTGES O14684 1/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
SYK P43405 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377580 0.81 GSK3B (0.87) GSK3BMAPTDYRK1ACDC7DBF4
SCHEMBL5381452 0.80 GSK3B (0.65) GSK3BIDO1CYP19A1CDC7DBF4
SCHEMBL5380569 0.79 GSK3B (0.73) GSK3BMAPTDYRK1ACDC7DBF4
SCHEMBL5375235 0.79 IDO1 (0.49) GSK3BIDO1MAPTCYP19A1DYRK1A
SCHEMBL5381549 0.76 GSK3B (1.00) GSK3BMAPTPOLBCDC7DBF4
SCHEMBL5391583 0.75 GSK3B (0.67) GSK3BCDC7RAB9AMAPK13MAPK12
SCHEMBL5380875 0.75 GSK3B (0.75) GSK3BMAPTDYRK1ACDC7DBF4
SCHEMBL5400000 0.73 GSK3B (0.73) GSK3BMAPTCDC7MAPK13MAPK12
SCHEMBL5381426 0.73 GSK3B (0.78) GSK3BMAPTCYP19A1POLBCDC7
SCHEMBL5384096 0.73 GSK3B (0.73) GSK3BRAB9AMAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed