SCHEMBL5375235

SCHEMBL5375235

COc1cc(-c2cc(=O)nc(-c3ccncc3)[nH]2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
CLK1 P49759 1/20 0.46
PKN1 Q16512 1/20 0.44
PKN2 Q16513 1/20 0.44
MAPT P10636 1/20 0.43
DYRK1A Q13627 1/20 0.41
MAPK13 O15264 3/20 0.40
MAPK12 P53778 3/20 0.40
MAPK11 Q15759 3/20 0.40
MAPK14 Q16539 3/20 0.40
CYP19A1 P11511 1/20 0.40
LRRK2 Q5S007 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
GRIA1 P42261 2/20 0.38
GRIA2 P42262 2/20 0.38
GRIA3 P42263 2/20 0.38
GRIA4 P48058 2/20 0.38
GSK3B P49841 1/20 0.38
RAF1 P04049 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377577 0.81 CDC7 (0.49) IDO1PKN1PKN2MAPTDYRK1A
SCHEMBL5381446 0.80 GSK3B (0.47) IDO1MAPTMAPK13MAPK12MAPK11
SCHEMBL5375238 0.79 GSK3B (0.60) IDO1PKN1PKN2MAPTDYRK1A
SCHEMBL5381545 0.76 CDC7 (0.59) IDO1PKN1PKN2MAPTMAPK13
SCHEMBL5391579 0.75 MAPK14 (0.56) MAPK13MAPK12MAPK11MAPK14NPC1
SCHEMBL5380873 0.73 MAPK14 (0.49) MAPTMAPK13MAPK12MAPK11MAPK14
SCHEMBL5384093 0.73 GCGR (0.56) MAPK13MAPK12MAPK11MAPK14NPC1
SCHEMBL5399995 0.73 MAPK14 (0.54) MAPK13MAPK12MAPK11MAPK14GSK3B
SCHEMBL7395689 0.73 MAPK14 (0.48) MAPTMAPK13MAPK12MAPK11MAPK14
SCHEMBL5383550 0.73 CDC7 (0.53) MAPK14NPC1RAB9ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed