SCHEMBL5376058

SCHEMBL5376058

O=CCCC#Cc1cccnc1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 5/20 0.58
CHRNA4 P43681 5/20 0.58
CYP2A6 P11509 5/20 0.57
CYP2C9 P11712 3/20 0.57
CYP2B6 P20813 3/20 0.57
CYP2C19 P33261 3/20 0.57
CYP2E1 P05181 2/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2D6 P10635 2/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2C8 P10632 1/20 0.56
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
ERN1 O75460 1/20 0.43
FFAR1 O14842 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28415042 0.83 CYP2A6 (0.61) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL5376053 0.81 CHRNB2 (0.63) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL3044684 0.79 CHRNB2 (0.70) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL10453306 0.78 CYP1A2 (0.48) CYP2C9CYP2C19CYP3A4CYP1A2FFAR1
SCHEMBL4065112 0.77 CHRNB2 (0.63) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL14085349 0.77 CYP2A6 (0.73) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL14085289 0.77 CHRNB2 (0.69) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL5032508 0.75 CHRNB2 (0.59) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL1841748 0.75 CHRNB2 (0.64) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL3673693 0.75 CHRNB2 (0.69) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253169-B2 Aza compounds, pharmaceutical compositions and methods of use GLIAMED, INC. (US) 2007-08-07 US disclosed