SCHEMBL5377385

SCHEMBL5377385

O=c1ccc(Cc2ccc(Cl)c(Oc3cccc(F)c3)c2)n[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.54
AKR1B1 P15121 3/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
SLC6A4 P31645 3/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34
KCNH2 Q12809 1/20 0.34
FFAR1 O14842 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
DRD4 P21917 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
ERBB3 P21860 1/20 0.33
ERBB4 Q15303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381993 0.90 CYP3A4 (0.47) CYP3A4AKR1B1SLC6A4HTR2AKCNH2
SCHEMBL5365181 0.89 CYP3A4 (0.67) CYP3A4AKR1B1FNTAFNTBPGGT1B
SCHEMBL4367667 0.88 CYP3A4 (0.53) CYP3A4AKR1B1THRATHRBCYP2C9
SCHEMBL5364926 0.87 CYP3A4 (0.54) CYP3A4FNTAFNTBPGGT1BSLC6A4
SCHEMBL5365245 0.87 CYP3A4 (0.49) CYP3A4FNTAFNTBPGGT1BPRMT5
SCHEMBL5376942 0.87 CYP3A4 (0.54) CYP3A4SLC6A4HTR2AKCNH2CYP2C9
SCHEMBL5385700 0.87 CYP3A4 (0.54) CYP3A4THRATHRBADORA2AADORA1
SCHEMBL5365375 0.86 CYP3A4 (0.52) CYP3A4AKR1B1SLC6A4HTR2AKCNH2
SCHEMBL5373776 0.85 CYP3A4 (0.43) CYP3A4AKR1B1THRATHRBCYP2C9
SCHEMBL5377579 0.84 CYP3A4 (0.52) CYP3A4FNTAFNTBPGGT1BPRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed