SCHEMBL5365375

SCHEMBL5365375

O=c1ccc(Cc2ccc(Cl)c(Oc3cccc(C(F)(F)F)c3)c2)n[nH]1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.52
AKR1B1 P15121 2/20 0.42
KIF11 P52732 1/20 0.38
HTR2A P28223 3/20 0.37
SLC6A4 P31645 3/20 0.37
KCNH2 Q12809 3/20 0.37
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
EGFR P00533 2/20 0.36
ERBB2 P04626 2/20 0.36
BRAF P15056 1/20 0.36
ERBB3 P21860 1/20 0.36
ERBB4 Q15303 1/20 0.36
ICAM1 P05362 1/20 0.36
SELE P16581 1/20 0.36
FAAH O00519 1/20 0.36
STK39 Q9UEW8 1/20 0.36
DDR1 Q08345 1/20 0.35
P2RY1 P47900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365456 0.89 CYP3A4 (0.50) CYP3A4AKR1B1KIF11ALDH1A1POLB
SCHEMBL5377299 0.88 CYP3A4 (0.47) CYP3A4AKR1B1KIF11ALDH1A1POLB
SCHEMBL5377385 0.86 CYP3A4 (0.54) CYP3A4AKR1B1HTR2ASLC6A4KCNH2
SCHEMBL5365181 0.86 CYP3A4 (0.67) CYP3A4AKR1B1HTR2ASLC6A4KCNH2
SCHEMBL4367667 0.85 CYP3A4 (0.53) CYP3A4AKR1B1
SCHEMBL5364926 0.84 CYP3A4 (0.54) CYP3A4HTR2ASLC6A4KCNH2ICAM1
SCHEMBL5385700 0.84 CYP3A4 (0.54) CYP3A4POLBFAAHSTK39
SCHEMBL5376942 0.84 CYP3A4 (0.54) CYP3A4HTR2ASLC6A4KCNH2POLB
SCHEMBL5374482 0.82 CYP3A4 (0.61) CYP3A4AKR1B1HTR2ASLC6A4KCNH2
SCHEMBL5377579 0.82 CYP3A4 (0.52) CYP3A4HTR2ASLC6A4KCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed