SCHEMBL5377456

SCHEMBL5377456

O=C(/C=C1/c2ccccc2NCCC1(F)F)NC[C@@H](O)CO

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.35
CNR2 P34972 1/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
AVPR2 P30518 12/20 0.32
AVPR1A P37288 7/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
MAP2K2 P36507 1/20 0.32
MAP2K1 Q02750 1/20 0.32
PRKCZ Q05513 1/20 0.32
IARS2 Q9NSE4 1/20 0.32
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377463 1.00 SLC6A2 (0.35) SLC6A2CNR2KDM4EALDH1A1HPGD
SCHEMBL5395013 1.00 SLC6A2 (0.35) SLC6A2CNR2KDM4EALDH1A1HPGD
SCHEMBL5395019 1.00 SLC6A2 (0.35) SLC6A2CNR2KDM4EALDH1A1HPGD
SCHEMBL3807603 0.78 AVPR2 (0.51) KDM4EALDH1A1AVPR2AVPR1ACYP3A4
SCHEMBL3807598 0.78 AVPR2 (0.51) KDM4EALDH1A1AVPR2AVPR1ACYP3A4
SCHEMBL3557117 0.76 AVPR2 (0.35) KDM4EALDH1A1HPGDAVPR2AVPR1A
SCHEMBL3557118 0.76 AVPR2 (0.35) KDM4EALDH1A1HPGDAVPR2AVPR1A
SCHEMBL7680383 0.76 CYP2C19 (0.45) KDM4EALDH1A1HPGDCYP3A4CYP2C19
SCHEMBL14590035 0.75 TGM2 (0.44) KDM4EALDH1A1AVPR2AVPR1A
SCHEMBL14590031 0.75 ALDH1A1 (0.34) KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183271-B2 4,4-difluoro-1,2,3,4-tetrahydro-5h-1-benzazepine derivative or salt thereof ASTELLAS PHARMA INC. (JP) 2007-02-27 US claimed