SCHEMBL5370543

SCHEMBL5370543

COc1ccc(Cc2ccc(=O)[nH]n2)cc1Oc1cccc(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
AR P10275 3/20 0.42
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
FNTA P49354 2/20 0.39
FNTB P49356 2/20 0.39
PGGT1B P53609 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
P2RX3 P56373 4/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
EPAS1 Q99814 3/20 0.36
VEGFA P15692 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5375295 0.89 CYP3A4 (0.47) CYP3A4ARCYP2C9CYP2C19FNTA
SCHEMBL5382226 0.89 CACNA1G (0.44) CYP3A4ARCYP2C9TSHRCYP2C19
SCHEMBL5377579 0.87 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19FNTAFNTB
SCHEMBL5374410 0.87 CYP3A4 (0.49) CYP3A4FNTAFNTBPGGT1BP2RX3
SCHEMBL5370328 0.87 CYP3A4 (0.47) CYP3A4FNTAFNTBPGGT1BP2RX3
SCHEMBL5365424 0.85 CYP3A4 (0.48) CYP3A4CYP2C9TSHRCYP2C19SMN1; SMN2
SCHEMBL5373732 0.84 CYP3A4 (0.45) CYP3A4ARCYP2C9CYP2C19FNTA
SCHEMBL5372848 0.80 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19PRMT5WDR77
SCHEMBL14570721 0.79 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19SMN1; SMN2EPAS1
SCHEMBL5368948 0.79 CYP3A4 (0.75) CYP3A4FNTAFNTBPGGT1BP2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed