SCHEMBL5377729

SCHEMBL5377729

O=C(c1c(F)cccc1F)c1cc(Cc2ccc(=O)[nH]n2)cc2ccoc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.72
PARP1 P09874 4/20 0.35
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
PSMB11 A5LHX3 1/20 0.31
PSMA7 O14818 1/20 0.31
PSMB1 P20618 1/20 0.31
PSMA1 P25786 1/20 0.31
PSMA2 P25787 1/20 0.31
PSMA3 P25788 1/20 0.31
PSMA4 P25789 1/20 0.31
PSMB8 P28062 1/20 0.31
PSMB9 P28065 1/20 0.31
PSMA5 P28066 1/20 0.31
PSMB4 P28070 1/20 0.31
PSMB6 P28072 1/20 0.31
PSMB5 P28074 1/20 0.31
PSMB10 P40306 1/20 0.31
PSMB3 P49720 1/20 0.31
PSMB2 P49721 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365374 0.91 CYP3A4 (0.68) CYP3A4PARP1THRATHRBPSMB11
SCHEMBL5373725 0.86 CYP3A4 (0.80) CYP3A4PARP1THRATHRBCFD
SCHEMBL5372475 0.84 CYP3A4 (1.00) CYP3A4PARP1AKR1B1PKM
SCHEMBL5368780 0.83 CYP3A4 (0.74) CYP3A4PARP1THRATHRBAKR1B1
SCHEMBL5368514 0.82 CYP3A4 (0.80) CYP3A4THRATHRBTDP1
SCHEMBL5365060 0.82 CYP3A4 (0.71) CYP3A4THRATHRBAKR1B1
SCHEMBL5368912 0.82 CYP3A4 (0.83) CYP3A4PARP1THRATHRBAKR1B1
SCHEMBL5371101 0.82 CYP3A4 (0.75) CYP3A4PKM
SCHEMBL5368824 0.81 CYP3A4 (0.70) CYP3A4AKR1B1
SCHEMBL5377033 0.80 CYP3A4 (0.76) CYP3A4THRATHRBAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed