SCHEMBL5368912

SCHEMBL5368912

O=C(c1cc(Cl)cc(Cl)c1)c1cc(Cc2ccc(=O)[nH]n2)cc2ccoc12

nearest known ligand 0.83

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.83
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
AKR1B1 P15121 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368514 0.92 CYP3A4 (0.80) CYP3A4THRATHRB
SCHEMBL5372475 0.91 CYP3A4 (1.00) CYP3A4AKR1B1PARP1
SCHEMBL5373725 0.87 CYP3A4 (0.80) CYP3A4THRATHRBPARP1
SCHEMBL5377033 0.87 CYP3A4 (0.76) CYP3A4THRATHRBAKR1B1
SCHEMBL5368780 0.86 CYP3A4 (0.74) CYP3A4THRATHRBAKR1B1PARP1
SCHEMBL5365060 0.85 CYP3A4 (0.71) CYP3A4THRATHRBAKR1B1
SCHEMBL5375137 0.83 CYP3A4 (0.67) CYP3A4THRATHRB
SCHEMBL5369076 0.83 CYP3A4 (0.67) CYP3A4THRATHRBPARP1
SCHEMBL5367220 0.83 CYP3A4 (0.84) CYP3A4THRATHRBAKR1B1
SCHEMBL5377729 0.82 CYP3A4 (0.72) CYP3A4THRATHRBAKR1B1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed