SCHEMBL5368780

SCHEMBL5368780

O=C(c1ccccc1Cl)c1cc(Cc2ccc(=O)[nH]n2)cc2ccoc12

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.74
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 3/20 0.32
RORB Q92753 1/20 0.32
RECQL P46063 1/20 0.32
MAPK7 Q13164 1/20 0.32
VNN1 O95497 1/20 0.32
POLB P06746 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
PARP1 P09874 1/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
IGFBP3 P17936 1/20 0.31
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
AKR1B1 P15121 1/20 0.31
KMT2A Q03164 1/20 0.31
CCNA2 P20248 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377033 0.89 CYP3A4 (0.76) CYP3A4CYP1A2CYP2C19ALDH1A1POLB
SCHEMBL5365374 0.88 CYP3A4 (0.68) CYP3A4ALDH1A1MAPK7VNN1PARP1
SCHEMBL5373725 0.88 CYP3A4 (0.80) CYP3A4CYP1A2ALDH1A1POLBPARP1
SCHEMBL5368514 0.86 CYP3A4 (0.80) CYP3A4CYP1A2CYP2C19ALDH1A1VNN1
SCHEMBL5368912 0.86 CYP3A4 (0.83) CYP3A4PARP1THRATHRBAKR1B1
SCHEMBL5372475 0.85 CYP3A4 (1.00) CYP3A4CYP2C19ALDH1A1VNN1PARP1
SCHEMBL5377729 0.83 CYP3A4 (0.72) CYP3A4PARP1THRATHRBAKR1B1
SCHEMBL5365060 0.82 CYP3A4 (0.71) CYP3A4ALDH1A1POLBTHRATHRB
SCHEMBL5369076 0.79 CYP3A4 (0.67) CYP3A4ALDH1A1VNN1POLBPARP1
SCHEMBL5375137 0.79 CYP3A4 (0.67) CYP3A4CYP1A2POLBKDM4ETHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed