SCHEMBL537820

SCHEMBL537820

CC(C)(O)c1ccc2c(n1)CCCC2

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 5/20 0.45
ADRA2B P18089 5/20 0.45
ADRA2C P18825 5/20 0.45
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SORT1 Q99523 2/20 0.36
CDK5 Q00535 3/20 0.33
CDK5R1 Q15078 3/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALOX15 P16050 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857053 0.85 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL12744626 0.83 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL21107870 0.83 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL21107629 0.83 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL20877628 0.83 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL24378402 0.83 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL18806199 0.81 ADRA2A (0.40) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL21451248 0.79 ADRA2A (0.39) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL12942916 0.77 ADRA2A (0.38) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL29875556 0.73 SORT1 (0.40) ADRA2AADRA2BADRA2CHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215054-B8 AMIDE DERIVATIVES AS ION-CHANNEL LIGANDS AND PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME EVOTEC AG (DE) 2012-02-08 EP disclosed