SCHEMBL5378232

SCHEMBL5378232

O=C(NCC1CN(C(=O)OCc2ccc(F)cc2F)CCO1)c1ccc(O)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 5/20 0.48
ENPP2 Q13822 2/20 0.43
ACKR3 P25106 1/20 0.42
NAMPT P43490 3/20 0.42
BCL9 O00512 1/20 0.41
CTNNB1 P35222 1/20 0.41
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425365 1.00 GRIN2B (0.48) GRIN2BENPP2ACKR3NAMPTBCL9
SCHEMBL5360981 0.90 ENPP2 (0.42) GRIN2BENPP2HPGDALDH1A1KMT2A
SCHEMBL14425370 0.90 ENPP2 (0.42) GRIN2BENPP2HPGDALDH1A1KMT2A
SCHEMBL14425360 0.89 GRIN2B (0.47) GRIN2BENPP2NAMPTGAAHPGD
SCHEMBL5365350 0.89 GRIN2B (0.47) GRIN2BENPP2NAMPTGAAHPGD
SCHEMBL14425314 0.87 F2 (0.48) GRIN2BENPP2NAMPTCYP1A2GAA
SCHEMBL5362085 0.87 F2 (0.48) GRIN2BENPP2NAMPTCYP1A2GAA
SCHEMBL14425445 0.87 F2 (0.48) GRIN2BENPP2NAMPTCYP1A2GAA
SCHEMBL5364450 0.85 GRIN2B (0.48) GRIN2BENPP2NAMPTCYP1A2GAA
SCHEMBL14425359 0.85 GRIN2B (0.48) GRIN2BENPP2NAMPTCYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed