SCHEMBL5378409

SCHEMBL5378409

Cc1nc(-c2ccccc2)c(-c2ccccc2)n1CCCCCCCC(=O)O

nearest known ligand 0.78

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FAAH O00519 15/20 0.78
CNR1 P21554 1/20 0.58
CNR2 P34972 1/20 0.58
PLA2G4A P47712 1/20 0.58
PTGIR P43119 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370606 1.00 FAAH (0.78) FAAHCNR1CNR2PLA2G4APTGIR
SCHEMBL14502383 1.00 FAAH (0.78) FAAHCNR1CNR2PLA2G4APTGIR
SCHEMBL5366194 0.89 FAAH (0.76) FAAHCNR1CNR2PLA2G4A
SCHEMBL8113624 0.88 FAAH (0.61) FAAHPTGIR
SCHEMBL8103885 0.88 FAAH (0.61) FAAHPTGIR
SCHEMBL8104725 0.88 FAAH (0.61) FAAHPTGIR
SCHEMBL8104252 0.88 FAAH (0.61) FAAHPTGIR
SCHEMBL5384210 0.87 FAAH (0.80) FAAHCNR1CNR2PLA2G4A
SCHEMBL5388273 0.87 FAAH (0.80) FAAHCNR1CNR2PLA2G4A
SCHEMBL5387755 0.87 FAAH (0.80) FAAHCNR1CNR2PLA2G4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39634-E1 Bisarylimidazoly fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-15 US disclosed
US-RE39634-E1 Bisarylimidazoly fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-15 US disclosed
US-RE39634-E1 Bisarylimidazoly fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-15 US disclosed
EP-1389107-A4 BISARYLIMIDAZOLYL FATTY ACID AMIDE HYDROLASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2005-10-12 EP disclosed
EP-1389107-A1 BISARYLIMIDAZOLYL FATTY ACID AMIDE HYDROLASE INHIBITORS Bristol-Myers Squibb Company (US) 2004-02-18 EP disclosed
US-6562846-B2 Bisarylimidazolyl fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2003-05-13 US disclosed
US-20020188009-A1 Bisarylimidazolyl fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2002-12-12 US disclosed
WO-2002087569-A1 BISARYLIMIDAZOLYL FATTY ACID AMIDE HYDROLASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2002-11-07 WO disclosed
EP-0626969-B1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORP (US) 2000-05-24 EP disclosed
US-5663053-A COENZYME A TRANSACYLASE FOR SCREENING SMITHKLINE BEECHAM CORPORATION (US) 1997-09-02 US disclosed
US-5648373-A CoA-IT and PAF inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1997-07-15 US disclosed
EP-0626969-A4 CoA-IT AND PAF INHIBITORS. SMITHKLINE BEECHAM CORP (US) 1995-04-19 EP disclosed
EP-0626969-A1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-12-07 EP disclosed
WO-1993016674-A1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-09-02 WO disclosed
EP-0550502-A1 SUBSTITUTED IMIDAZOLES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-07-14 EP disclosed
WO-1992004330-A1 SUBSTITUTED IMIDAZOLES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-03-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020188009-A1 Bisarylimidazolyl fatty acid amide hydrolase inhibitors FAAH, FAAH2, FASN FAAH 1/4885CNR1 172/4885CNR2 102/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.