SCHEMBL5380506

SCHEMBL5380506

Nc1ccccc1N(C(=O)c1ccc(Cn2c(=S)n(-c3ccccc3)c3ccccc32)cc1)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PGR P06401 1/20 0.32
CCR2 P41597 1/20 0.32
KLK1 P06870 1/20 0.31
APEX1 P27695 1/20 0.31
MITF O75030 1/20 0.31
HTT P42858 1/20 0.31
BACE1 P56817 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC2 Q92769 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5380499 0.83 PTAFR (0.39) HDAC1KDM4EMAPTKMT2AMEN1
SCHEMBL3539202 0.76 HDAC1 (0.57) HDAC1HDAC10HDAC6HDAC3HDAC2
SCHEMBL5611501 0.70 CYP1A2 (0.46) HDAC1KDM4ESMN1; SMN2HDAC10HDAC6
SCHEMBL10055041 0.69 ALDH1A1 (0.49) HDAC1KDM4EMAPTKMT2AMEN1
SCHEMBL3540141 0.65 HDAC1 (0.63) HDAC1HDAC10HDAC6HDAC3HDAC2
SCHEMBL10453089 0.63 ESR1 (0.49) HDAC1KMT2AMEN1HDAC10HDAC6
SCHEMBL2362869 0.62 HDAC1 (0.54) HDAC1KMT2AMEN1HDAC10HDAC6
SCHEMBL16684997 0.61 POLB (0.47) KDM4EMAPTKMT2ASMN1; SMN2TDP1
SCHEMBL9767715 0.61 CES2 (0.50) MAPTKMT2ASMN1; SMN2HTTBACE1
SCHEMBL27482363 0.61 CA1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824831-A2 HISTONE DEACETYLASE INHIBITORS Takeda San Diego, Inc. (US) 2007-08-29 EP disclosed
WO-2006066133-A2 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed