SCHEMBL5380666

SCHEMBL5380666

CCCc1c(CO)cnn1Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
MAPK14 Q16539 1/20 0.43
RECQL P46063 1/20 0.43
CYP19A1 P11511 1/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 3/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
HTT P42858 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37
BRD4 O60885 1/20 0.37
AADAT Q8N5Z0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31584017 0.88 PTGDR2 (0.47) TSHRRECQLALDH1A1POLBPTGDR2
SCHEMBL2820258 0.82 NPBWR1 (0.41) ALDH1A1PTGDR2BRD4
SCHEMBL23400358 0.82 TSHR (0.46) TSHRMAPK14RECQLCYP19A1ALDH1A1
SCHEMBL21332896 0.78 TSHR (0.53) TSHRRECQLALDH1A1POLBPTGDR2
SCHEMBL7592930 0.77 ALDH1A1 (0.52) TSHRMAPK14RECQLCYP19A1ALDH1A1
SCHEMBL26042 0.76 NR4A3 (0.54) MAPK14ALDH1A1POLB
SCHEMBL5377123 0.75 TSHR (0.43) TSHRMAPK14RECQLCYP19A1ALDH1A1
SCHEMBL5381957 0.74 RECQL (0.46) TSHRRECQLCYP19A1ALDH1A1HSD17B10
SCHEMBL25342354 0.73 ALDH1A1 (0.48) TSHRALDH1A1HTTHSD17B10
SCHEMBL5382860 0.73 SMN1; SMN2 (0.58) TSHRMAPK14CYP19A1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179823-B1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-20 US disclosed
EP-1457490-A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity Takeda Chemical Industries, Ltd. (JP) 2004-09-15 EP disclosed
EP-1228067-B1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-07-14 EP disclosed