SCHEMBL5383591

SCHEMBL5383591

O=c1cc(-c2ccnc(Cl)c2)[nH]c(CCCc2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.50
HCAR2 Q8TDS4 4/20 0.43
MAPKAPK2 P49137 3/20 0.43
CDC7 O00311 1/20 0.43
ROCK2 O75116 1/20 0.43
MAP4K4 O95819 1/20 0.43
CDK2 P24941 1/20 0.43
HIPK2 Q9H2X6 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43
DAO P14920 1/20 0.40
IDO1 P14902 1/20 0.40
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5375436 0.84 GSK3B (0.48) GSK3BHCAR2MAPKAPK2DAOGPR84
SCHEMBL5387928 0.84 GSK3B (0.65) GSK3BHCAR2CDC7DAOMAPK13
SCHEMBL5382154 0.83 GSK3B (0.47) GSK3BHCAR2MAPKAPK2DAOIDO1
SCHEMBL5383593 0.81 GSK3B (0.72) GSK3BHCAR2DAOMAPK13MAPK12
SCHEMBL5386067 0.78 GSK3B (0.51) GSK3BHCAR2DAO
SCHEMBL5390682 0.76 GSK3B (0.64) GSK3BCDC7DAOTUBB4ATUBB
SCHEMBL5390574 0.76 GSK3B (0.49) GSK3BHCAR2DAOTUBB4ATUBB
SCHEMBL5381446 0.70 GSK3B (0.47) GSK3BMAPKAPK2CDC7ROCK2MAP4K4
SCHEMBL5376093 0.70 GSK3B (0.63) GSK3BMAPKAPK2CDC7CDK2DAO
SCHEMBL12318506 0.69 NPC1 (0.58) GSK3BMAPKAPK2CDC7ROCK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed