SCHEMBL5384802

SCHEMBL5384802

CCOC(=O)c1cn(Cc2ccc(Oc3ccccc3)cc2)nc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LMNA P02545 1/20 0.49
MAP2K1 Q02750 2/20 0.45
TSHR P16473 2/20 0.44
KDM4E B2RXH2 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KLKB1 P03952 1/20 0.44
CRHBP P24387 2/20 0.43
CRHR2 Q13324 2/20 0.43
KMT2A Q03164 1/20 0.43
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
AGTR1 P30556 1/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852276 0.90 ALDH1A1 (0.59) ALDH1A1LMNATSHRKDM4ENPC1
SCHEMBL5377176 0.84 ALDH1A1 (0.46) ALDH1A1LMNAMAP2K1TSHRKDM4E
SCHEMBL5385889 0.78 FFAR1 (0.57)
SCHEMBL5385608 0.78 MAPK1 (0.54) ALDH1A1LMNANPC1RAB9AKLKB1
SCHEMBL4851123 0.78 ALDH1A1 (0.49) ALDH1A1LMNATSHRKDM4ENPC1
SCHEMBL4544356 0.77 ALDH1A1 (0.57) ALDH1A1LMNATSHRKDM4ENPC1
SCHEMBL5372048 0.76 MEN1 (0.51) ALDH1A1LMNATSHRKMT2AL3MBTL1
SCHEMBL1052418 0.76 PDE4D (0.49) ALDH1A1LMNAKDM4ENPC1KMT2A
SCHEMBL20477440 0.76 ALDH1A1 (0.56) ALDH1A1LMNATSHRKDM4ECRHBP
SCHEMBL20477455 0.76 LMNA (0.56) ALDH1A1LMNATSHRKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179823-B1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-20 US disclosed
EP-1457490-A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity Takeda Chemical Industries, Ltd. (JP) 2004-09-15 EP disclosed
EP-1228067-B1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-07-14 EP disclosed
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed