SCHEMBL5386532

SCHEMBL5386532

CCOc1cccc(-c2nc(-c3ccncc3)cc(=O)[nH]2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.62
S1PR1 P21453 2/20 0.51
KDM4E B2RXH2 2/20 0.48
MAPT P10636 2/20 0.48
GAA P10253 1/20 0.48
THRB P10828 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.44
TP53 P04637 2/20 0.44
ROCK2 O75116 2/20 0.43
ROCK1 Q13464 2/20 0.43
NPC1 O15118 1/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5391583 0.86 GSK3B (0.67) GSK3BNPC1RAB9AMAPK13RAF1
SCHEMBL5386526 0.81 S1PR1 (0.51) GSK3BS1PR1KDM4EMAPTGAA
SCHEMBL5383553 0.80 GSK3B (0.72) GSK3BNPC1RAB9AMAPK14
SCHEMBL5381549 0.78 GSK3B (1.00) GSK3BMAPTGAASMN1; SMN2ALDH1A1
SCHEMBL5377580 0.77 GSK3B (0.87) GSK3BMAPTGAAROCK2ROCK1
SCHEMBL7391408 0.77 GSK3B (0.72) GSK3BKDM4EMAPTSMN1; SMN2TP53
SCHEMBL5392045 0.77 GSK3B (0.72) GSK3BGAAROCK2ROCK1NPC1
Hydrochloric Acid SCHEMBL5386672 0.75 GSK3B (0.61) GSK3BSMN1; SMN2ROCK2MAPK14
SCHEMBL5388178 0.74 GSK3B (0.67) GSK3BMAPK13RAF1MAPK12MAPK11
SCHEMBL5376063 0.74 GSK3B (0.76) GSK3BKDM4EMAPTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed