SCHEMBL5397278

SCHEMBL5397278

N#CC1(NC(=O)[C@H](CS(=O)(=O)Cc2ccccc2)NCC(F)(F)c2cccs2)CC1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 17/20 0.57
CTSS P25774 16/20 0.57
CTSB P07858 13/20 0.57
CTSK P43235 11/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5392764 0.83 CTSL (0.48) CTSLCTSSCTSBCTSK
SCHEMBL2820824 0.81 CTSL (0.71) CTSLCTSSCTSBCTSK
SCHEMBL2820825 0.81 CTSL (0.71) CTSLCTSSCTSBCTSK
SCHEMBL2820828 0.81 CTSL (0.71) CTSLCTSSCTSBCTSK
SCHEMBL2820741 0.80 CTSS (0.59) CTSLCTSSCTSBCTSK
SCHEMBL2820743 0.80 CTSS (0.59) CTSLCTSSCTSBCTSK
SCHEMBL2821047 0.77 CTSL (0.89) CTSLCTSSCTSBCTSK
SCHEMBL2822122 0.77 CTSL (0.71) CTSLCTSSCTSBCTSK
SCHEMBL2822120 0.77 CTSL (0.71) CTSLCTSSCTSBCTSK
SCHEMBL2821048 0.77 CTSL (0.89) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007505920-A 2007-03-15 JP claimed
EP-1663958-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2006-06-07 EP claimed
WO-2005028429-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-03-31 WO claimed
EP-1663958-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2006-06-07 EP disclosed
WO-2005028429-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-03-31 WO disclosed