SCHEMBL5398

SCHEMBL5398

[CH2]c1nc2ccccc2[nH]1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
NPC1 O15118 3/20 0.60
RAB9A P51151 3/20 0.60
NPSR1 Q6W5P4 2/20 0.60
KDM4E B2RXH2 2/20 0.60
PKM P14618 2/20 0.60
ABCB11 O95342 1/20 0.60
TP53 P04637 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
HSD17B10 Q99714 1/20 0.60
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
MASP2 O00187 1/20 0.56
NUDT1 P36639 1/20 0.56
AOC3 Q16853 1/20 0.56
GAA P10253 2/20 0.52
POLB P06746 2/20 0.50
IDO1 P14902 1/20 0.50
DDAH1 O94760 1/20 0.50
BCHE P06276 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7528714 0.92 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL4388269 0.76 KDM4E (0.55) ALDH1A1NPC1RAB9AKDM4EPKM
SCHEMBL172216 0.75 NPC1 (1.00) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL30561047 0.75 NPC1 (1.00) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL30634854 0.75 NPC1 (1.00) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL16403339 0.74 PLAUR (0.61) ALDH1A1NPC1RAB9ANPSR1KDM4E
Water SCHEMBL9817804 0.73 NPC1 (0.95) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL29034384 0.73 ALDH1A1 (0.62) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL9214713 0.73 ALDH1A1 (0.68) ALDH1A1NPC1RAB9ANPSR1KDM4E
SCHEMBL1705977 0.71 ALDH1A1 (0.60) ALDH1A1NPC1RAB9ANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2665 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12029739-B2 SHP2 inhibitor and use thereof KANAPH THERAPEUTICS INC. (KR) 2024-07-09 US claimed
US-20240189306-A1 SHP2 INHIBITOR AND USE THEREOF KANAPH THERAPEUTICS INC. (KR) 2024-06-13 US claimed
WO-2024104425-A1 KRAS INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 广东东阳光药业股份有限公司 2024-05-23 WO claimed
CN-118047801-A KRAS inhibitor compound, pharmaceutical composition and application thereof 广东东阳光药业股份有限公司 2024-05-17 CN claimed
EP-4368625-A1 SHP2 INHIBITOR AND USE THEREOF Kanaph Therapeutics Inc. (KR) 2024-05-15 EP claimed
CN-117916242-A SHP2 inhibitors and uses thereof 治纳辅医药科技有限公司 2024-04-19 CN claimed
CN-117551221-A Benzimidazolyl chitosan quaternary ammonium salt derivative and preparation and application thereof 中国科学院烟台海岸带研究所 2024-02-13 CN claimed
US-20240025892-A1 SALT INDUCIBLE KINASE INHIBITORS THE GENERAL HOSPITAL CORPORATION 2024-01-25 US claimed
CN-115043829-B Indole compound and preparation method and application thereof 河南农业大学 2023-07-25 CN claimed
EP-4192459-A1 SALT INDUCIBLE KINASE INHIBITORS The General Hospital Corporation (US) 2023-06-14 EP claimed
EP-0611375-A1 PEPTIDES INHIBITING IL-1 BETA RELEASE SANDOZ LTD. (CH) 1994-08-24 EP claimed
EP-0417555-B1 Pentamethine dyes and derivatives BAYER AG (DE) 1993-11-03 EP claimed
WO-1993009135-A1 PEPTIDES INHIBITING IL-1 BETA RELEASE SANDOZ LTD. (CH) 1993-05-13 WO claimed
US-5118814-A Pressure sensitive and heat sensitive recording media BAYER AKTIENGESELLSCHAFT (DE) 1992-06-02 US claimed
EP-0217256-B1 METHOD FOR QUENCHING FLUORESCENCE, AND CATIONIC DERIVATIVES OF NAPHTHALENE-PERI-DICARBOXAMIDE BAYER AG (DE) 1991-03-06 EP claimed
EP-0201221-B1 6-(1-ACYL-1-HYDROXY METHYL) PENICILLANIC ACID DERIVATIVES PFIZER INC. (US) 1990-08-01 EP claimed
EP-0370198-A1 Tetraindolyl heptamethine derivatives BAYER AG (DE) 1990-05-30 EP claimed
EP-0217256-A2 Method for quenching fluorescence, and cationic derivatives of naphthalene-peri-dicarboxamide BAYER AG (DE) 1987-04-08 EP claimed
EP-0173377-A2 Pyrimidone compounds, their preparation and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1986-03-05 EP claimed
EP-0086647-A2 Pyrimidone compounds, their preparation, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1983-08-24 EP claimed