SCHEMBL5403798

SCHEMBL5403798

COC1=Cc2ncn(-c3cc(OCc4ccccc4C(F)(F)F)c(C#N)s3)c2CC1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 13/20 0.62
IKBKE Q14164 8/20 0.62
TBK1 Q9UHD2 1/20 0.46
NEK2 P51955 4/20 0.44
CSF1R P07333 3/20 0.44
KDR P35968 3/20 0.44
LIMK1 P53667 3/20 0.44
STK3 Q13188 3/20 0.44
DYRK1A Q13627 3/20 0.44
BRSK1 Q8TDC3 3/20 0.44
PLK3 Q9H4B4 3/20 0.44
CLK4 Q9HAZ1 3/20 0.44
MAP4K5 Q9Y4K4 3/20 0.44
PLK4 O00444 2/20 0.44
AURKA O14965 2/20 0.44
JAK2 O60674 2/20 0.44
LCK P06239 2/20 0.44
FGFR1 P11362 2/20 0.44
SRC P12931 2/20 0.44
FLT1 P17948 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5399856 0.92 IKBKE (0.62) PLK1IKBKETBK1NEK2CSF1R
SCHEMBL5410566 0.88 IKBKE (0.66) PLK1IKBKETBK1NEK2CSF1R
SCHEMBL5409630 0.86 IKBKE (0.64) PLK1IKBKETBK1
SCHEMBL5399351 0.85 IKBKE (0.63) PLK1IKBKENEK2KDRPLK3
SCHEMBL5769049 0.84 IKBKE (0.44) PLK1IKBKETBK1
SCHEMBL5408899 0.84 IKBKE (0.41) PLK1IKBKETBK1
SCHEMBL5402250 0.82 IKBKE (0.41) PLK1IKBKETBK1CSF1RKIT
SCHEMBL5395239 0.82 IKBKE (0.43) PLK1IKBKETBK1
SCHEMBL5394634 0.81 IKBKE (0.45) PLK1IKBKETBK1
SCHEMBL5394828 0.81 IKBKE (0.42) PLK1IKBKETBK1CSF1RKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007522142-A 2007-08-09 JP claimed
EP-1720864-A1 BENZIMIDAZOL SUBSTITUTED THIOPHENE DERIVATIVES WITH ACTIVITY ON IKK3 GLAXO GROUP LIMITED (GB) 2006-11-15 EP claimed
WO-2005075465-A1 BENZIMIDAZOL SUBSTITUTED THIOPENE DERIVATIVES WITH ATCTIVITY ON IKK3 GLAXO GROUP LIMITED (GB) 2005-08-18 WO claimed