SCHEMBL540577

SCHEMBL540577

CC(=O)Nc1ncc(S(=O)(=O)Cl)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 8/20 0.43
CDK2 P24941 8/20 0.43
CDK4 P11802 4/20 0.43
CDK1 P06493 3/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
FFAR2 O15552 1/20 0.42
CCNE2 O96020 7/20 0.42
CCND1 P24385 3/20 0.42
CCNB2 O95067 2/20 0.42
CCNB1 P14635 2/20 0.42
CCNB3 Q8WWL7 2/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA3 P07451 2/20 0.41
CA4 P22748 2/20 0.41
CA6 P23280 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4860224 0.85 CCNE1 (0.44) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL27174909 0.85 FFAR2 (0.40) CCNE1CDK2LMNAMEN1KMT2A
SCHEMBL14419937 0.85 FFAR2 (0.52) CCNE1CDK2CDK4CDK1LMNA
Hydrochloric Acid SCHEMBL28108629 0.83 CCNE1 (0.43) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL6078335 0.83 CA2 (0.53) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL10154046 0.82 CA12 (0.54) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL15882463 0.82 CCNE1 (0.44) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL16731877 0.82 CCNE1 (0.49) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL10233482 0.81 OGA (0.45) CCNE1CDK2CDK4CDK1LMNA
SCHEMBL30760419 0.79 CA1 (0.49) CCNE1CDK2CDK4CDK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 167 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260092053-A1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2026-04-02 US disclosed
EP-4681774-A2 KHK INHIBITORS Gilead Sciences, Inc. (US) 2026-01-21 EP disclosed
EP-4313967-B1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2025-11-12 EP disclosed
US-12410160-B2 KHK inhibitors GILEAD SCIENCES, INC. (US) 2025-09-09 US disclosed
CN-115745910-B Chemical compound 安塔比奥公司 2025-05-27 CN disclosed
US-20240190860-A1 8-CYCLO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS LPA RECEPTOR 2 INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2024-06-13 US disclosed
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
EP-4313956-A1 8-CYCLO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS LPA RECEPTOR 2 INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2024-02-07 EP disclosed
EP-4073073-B1 THIENOPYRIMIDINE DERIVATIVES AS LPA RECEPTOR 2 INHIBITORS CHIESI FARM SPA (IT) 2023-12-06 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2007006760-A1 DICYCLOALKYL UREA GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2007-01-18 WO disclosed
WO-2007007886-A1 AN OXIME DERIVATIVE AND PREPARATIONS THEREOF MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-01-18 WO disclosed
WO-2007006814-A1 UREA GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2007-01-18 WO disclosed
EP-1723128-A1 HETEROARYL-UREAS AND THEIR USE AS GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2006-11-22 EP disclosed
US-20060183756-A1 Pyrrazolo-pyrimidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 2006-08-17 US disclosed
WO-2006084634-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-08-17 WO disclosed
WO-2005066145-A1 HETEROARYL-UREAS AND THEIR USE AS GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2005-07-21 WO disclosed
US-5360813-A Inhibitors of ergosterol biosynthesis J. URIACH & CIA. S.A. (ES) 1994-11-01 US disclosed
US-5344839-A Imidazole or triazole compounds J. URIACH & CIA. S.A. (ES) 1994-09-06 US disclosed
EP-0480215-A1 New sulfonamides as antifungal agents J. URIACH & CIA. S.A. (ES) 1992-04-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060183756-A1 Pyrrazolo-pyrimidine derivatives GRM1, GRM2, GRM3 CCNE1 2427/4885CDK2 506/4885CDK4 533/4885
US-20260092053-A1 KHK INHIBITORS KHK, SLC5A2, HK1 CCNE1 4317/4885CDK2 2411/4885CDK4 2297/4885
US-12410160-B2 KHK inhibitors KHK, KHDRBS1, NADK CCNE1 2915/4885CDK2 519/4885CDK4 1215/4885
US-20240190860-A1 8-CYCLO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS LPA RECEPTOR 2 INHIBITORS LPAR2, LPAR5, LPAR1 CCNE1 2107/4885CDK2 298/4885CDK4 1660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.