SCHEMBL541044

SCHEMBL541044

FNCc1cccc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.58
IDO1 P14902 2/20 0.56
HTR2A P28223 2/20 0.55
HTR2B P41595 2/20 0.55
HTR2C P28335 1/20 0.55
MLYCD O95822 1/20 0.54
ACP3 P15309 1/20 0.53
GAA P10253 2/20 0.53
MEN1 O00255 1/20 0.53
PLA2G1B P04054 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
ATG4B Q9Y4P1 1/20 0.53
MIF P14174 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
LMNA P02545 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4239980 0.88 DPP7 (0.59) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL46769 0.84 MLYCD (0.55) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL15129325 0.84 TAAR1 (0.55) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL29988585 0.84 MRGPRX4 (0.57) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL4368141 0.84 TAAR1 (0.59) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL42728 0.84 MRGPRX4 (0.57) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL18901273 0.84 TAAR1 (0.55) TAAR1IDO1HTR2AHTR2BHTR2C
Bromide SCHEMBL29093720 0.82 TAAR1 (0.53) TAAR1IDO1HTR2AHTR2BHTR2C
Hydrochloric Acid SCHEMBL8701788 0.82 IDO1 (0.54) TAAR1IDO1HTR2AHTR2BHTR2C
SCHEMBL4245195 0.82 DPP7 (0.55) TAAR1IDO1HTR2AHTR2BHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414346-A1 AUTOTAXIN INHIBITORS Merck Patent GmbH (DE) 2012-02-08 EP claimed
WO-2010112124-A1 AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-07 WO claimed
CN-108135168-A CCR2 modulators 凯莫森特里克斯股份有限公司 2018-06-08 CN disclosed
CN-105505128-B Near-infrared light response self-repairing coating and preparation method thereof 南京工业大学 2018-05-08 CN disclosed
CN-103102303-B As the benzyl amine derivative of CETP inhibitor DR. REDDY'S LABORATORIES LTD. (IN) 2015-10-28 CN disclosed
CN-104962543-A Oriented immobilization method for bacillus subtilis neutral protease UNIV SHANGHAI SCIENCE & TECH 2015-10-07 CN disclosed
CN-104151319-A Selective substituted pyridine ligands for neuronal nicotinic receptors ABBVIE INC 2014-11-19 CN disclosed
CN-103172562-A Trisubstituted amine compounds as inhibitors of cholesteryl ester transfer protein CETP TANABE SEIYAKU CO 2013-06-26 CN disclosed
EP-2440294-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS TRPM8 CHANNEL MODULATORS Janssen Pharmaceutica, N.V. (BE) 2012-04-18 EP disclosed
WO-2010144680-A1 BENZIMIDAZOLE DERIVATIVES USEFUL AS TRPM8 CHANNEL MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2010-12-16 WO disclosed
WO-2006103342-A9 INDANYL-PIPERAZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2007-10-25 WO disclosed