SCHEMBL543036

SCHEMBL543036

FC(F)(F)Oc1ccc([CH]Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
MAPT P10636 2/20 0.42
EPHX2 P34913 1/20 0.42
CYP2D6 P10635 1/20 0.41
KDM4E B2RXH2 2/20 0.40
MAOB P27338 1/20 0.40
AOC3 Q16853 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
GPR3 P46089 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
GRIK1 P39086 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2092050 0.81 PIM1 (0.49) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL13790221 0.81 CYP2D6 (0.50) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL254957 0.80 MAPT (0.56) PIM1PIM2MAPTEPHX2KDM4E
SCHEMBL15117409 0.79 PIM1 (0.47) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL28757636 0.77 MAPT (0.47) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL97114 0.77 ALDH1A1 (0.52) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL2116917 0.77 PIM1 (0.46) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL171790 0.77 ALDH1A1 (0.50) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL3396974 0.77 PIM1 (0.46) PIM1PIM2MAPTEPHX2CYP2D6
SCHEMBL1047423 0.77 PIM1 (0.46) PIM1PIM2MAPTEPHX2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414330-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS Merck Patent GmbH (DE) 2012-02-08 EP claimed
WO-2010115491-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-14 WO claimed