SCHEMBL5432012

SCHEMBL5432012

COc1cccc(Cn2cc(C3CC[N]C3c3ccc([N+](=O)[O-])cc3Cl)c3ccccc32)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 5/20 0.42
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC29A1 Q99808 1/20 0.38
SLC5A1 P13866 1/20 0.38
SLC5A2 P31639 1/20 0.38
SLC2A1 P11166 1/20 0.37
HTT P42858 1/20 0.37
CACNB4 O00305 1/20 0.37
CACNA1A O00555 1/20 0.37
CACNA1G O43497 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5441447 0.88 SLC2A1 (0.49) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL5800685 0.79 GRIN1 (0.41) MAPTSLC5A1SLC5A2SLC2A1POLB
SCHEMBL4858756 0.77 SLC2A1 (0.49) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL5434125 0.76 SLC5A1 (0.40) MAPTPDE4APDE4BPDE4CPDE4D
SCHEMBL5432493 0.73 SLC5A1 (0.42) ALDH1A1SMN1; SMN2LMNAMAPTSLC5A1
SCHEMBL5797794 0.68 SLC5A1 (0.46) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL4194784 0.66 MAPT (0.51) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL7032876 0.65 QPCT (0.56) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL13131367 0.65 MAPT (0.57) ALDH1A1KMT2ALMNAMAPTTP53
SCHEMBL5438268 0.65 CRHR1 (0.35) ALDH1A1SMN1; SMN2MAPTPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007501828-A 2007-02-01 JP claimed
EP-1654253-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2006-05-10 EP claimed
WO-2005019208-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2005-03-03 WO claimed
EP-1654253-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2006-05-10 EP disclosed
WO-2005019208-A1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES Grünenthal GmbH (DE) 2005-03-03 WO disclosed