SCHEMBL543284

SCHEMBL543284

O=C(OCc1cc(F)cc(C(F)(F)F)c1)N1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 6/20 0.47
ATXN2 Q99700 3/20 0.47
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TACR1 P25103 5/20 0.43
FFAR4 Q5NUL3 1/20 0.42
F13A1 P00488 1/20 0.41
TGM2 P21980 1/20 0.41
TGM1 P22735 1/20 0.41
TSHR P16473 2/20 0.41
CYP2D6 P10635 1/20 0.41
MGLL Q99685 1/20 0.41
HPGD P15428 2/20 0.40
CYP3A4 P08684 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
HTR2A P28223 1/20 0.40
ABAT P80404 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL543132 0.92 TACR1 (0.49) ENPP2ATXN2MEN1KMT2ATACR1
SCHEMBL28032625 0.86 ENPP2 (0.52) ENPP2ATXN2MEN1KMT2ATACR1
SCHEMBL543130 0.86 ENPP2 (0.55) ENPP2ATXN2MEN1KMT2ATACR1
SCHEMBL28032629 0.82 KMT2A (0.64) ENPP2ATXN2MEN1KMT2AHPGD
SCHEMBL543231 0.81 MEN1 (0.55) ENPP2ATXN2MEN1KMT2ATSHR
SCHEMBL542677 0.79 MEN1 (0.53) ENPP2ATXN2MEN1KMT2ATSHR
SCHEMBL16093830 0.79 ENPP2 (0.41) ENPP2ATXN2MEN1KMT2ATACR1
SCHEMBL543034 0.78 TACR1 (0.47) ENPP2ATXN2TACR1TSHRCYP2D6
SCHEMBL16093646 0.78 ENPP2 (0.40) ENPP2ATXN2TACR1FFAR4MGLL
SCHEMBL543075 0.77 DPP4 (0.42) ENPP2MEN1KMT2AF13A1TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414330-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS Merck Patent GmbH (DE) 2012-02-08 EP claimed
WO-2010115491-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-14 WO claimed