SCHEMBL545286

SCHEMBL545286

CN(Cc1ccc(N)cc1C(F)(F)F)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.47
CACNA1B Q00975 1/20 0.47
CACNA1C Q13936 1/20 0.47
NR1H2 P55055 2/20 0.40
GAA P10253 2/20 0.37
GLA P06280 1/20 0.37
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37
SLC6A4 P31645 4/20 0.36
HTR2C P28335 3/20 0.36
RXRA P19793 1/20 0.36
NR1H3 Q13133 1/20 0.36
PDK2 Q15119 1/20 0.35
POLQ O75417 3/20 0.35
SOS1 Q07889 1/20 0.35
HTR2A P28223 1/20 0.35
RIPK1 Q13546 1/20 0.34
ACHE P22303 1/20 0.34
EPHX2 P34913 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4655741 0.84 CACNA1G (0.46) CACNA1GCACNA1BCACNA1CNR1H2SLC6A4
SCHEMBL31468983 0.83 HTR2C (0.38) CACNA1GCACNA1BCACNA1CNR1H2SLC6A4
SCHEMBL8169426 0.83 RIPK1 (0.46) CACNA1GCACNA1BCACNA1CSLC6A4HTR2C
SCHEMBL5423901 0.82 NR1H2 (0.48) NR1H2GAAGLAPOLBTSHR
SCHEMBL13622928 0.82 HTR2C (0.37) CACNA1GCACNA1BCACNA1CNR1H2SLC6A4
SCHEMBL4656684 0.81 NOTUM (0.47) CACNA1GCACNA1BCACNA1CNR1H2GAA
SCHEMBL17705199 0.81 CACNA1G (0.36) CACNA1GCACNA1BCACNA1CNR1H2SLC6A4
SCHEMBL8162665 0.81 SLC6A4 (0.40) CACNA1GCACNA1BCACNA1CSLC6A4HTR2C
SCHEMBL20214469 0.81 CACNA1G (0.43) CACNA1GCACNA1BCACNA1CGAAPOLB
SCHEMBL18186254 0.80 HTR2C (0.38) CACNA1GCACNA1BCACNA1CNR1H2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110687-B2 Bicyclic compounds with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-07 US disclosed