SCHEMBL545297

SCHEMBL545297

CC(C)(C)N(Cc1ccc(N)cc1C(F)(F)F)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.46
GLA P06280 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
POLQ O75417 4/20 0.37
S1PR1 P21453 1/20 0.36
SLC6A4 P31645 6/20 0.36
SLC6A2 P23975 5/20 0.36
EPHX2 P34913 3/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
AR P10275 1/20 0.34
PPARG P37231 1/20 0.34
LMNA P02545 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL545287 0.86 NR1H2 (0.44) NR1H2GLAPOLBGAATSHR
SCHEMBL1818639 0.83 PTGDR2 (0.39) POLQS1PR1SLC6A4SLC6A2EPHX2
SCHEMBL5423901 0.83 NR1H2 (0.48) NR1H2GLAPOLBGAATSHR
SCHEMBL1438626 0.83 RIPK1 (0.41) TSHREPHX2MEN1KMT2AHTT
SCHEMBL15752820 0.81 PRKCI (0.38) POLBGAATSHREPHX2MEN1
SCHEMBL374610 0.79 NR1H2 (0.51) NR1H2GLAPOLBGAATSHR
SCHEMBL30401867 0.79 NR1H2 (0.51) NR1H2GLAPOLBGAATSHR
SCHEMBL15057213 0.78 SLC6A4 (0.42) TSHRSLC6A4SLC6A2EPHX2MEN1
SCHEMBL4937359 0.78 NR1H2 (0.48) NR1H2GLAPOLBGAATSHR
Hydrochloric Acid SCHEMBL16054675 0.77 NR1H2 (0.50) NR1H2GLAPOLBGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110687-B2 Bicyclic compounds with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-07 US disclosed