SCHEMBL545287

SCHEMBL545287

CC(C)(C)N(CCc1ccc(N)cc1C(F)(F)F)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.44
S1PR1 P21453 1/20 0.39
GLA P06280 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
POLQ O75417 5/20 0.36
EPHX2 P34913 4/20 0.34
AR P10275 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PPARG P37231 2/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SLC6A4 P31645 2/20 0.32
SLC6A2 P23975 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL545297 0.86 NR1H2 (0.46) NR1H2S1PR1GLAPOLBGAA
SCHEMBL31162543 0.77 NR1H2 (0.49) NR1H2GLAPOLBGAATSHR
SCHEMBL5423901 0.75 NR1H2 (0.48) NR1H2GLAPOLBGAATSHR
SCHEMBL28382816 0.75 NR1H2 (0.47) NR1H2S1PR1GLAPOLBGAA
SCHEMBL28851099 0.75 NR1H2 (0.47) NR1H2S1PR1GLAPOLBGAA
SCHEMBL1845384 0.74 MEN1 (0.46) EPHX2MEN1KMT2AHTTL3MBTL1
SCHEMBL4678727 0.73 EPHX2 (0.48) NR1H2GLAPOLBGAATSHR
SCHEMBL1205533 0.72 MAOA (0.49) TSHRMEN1KMT2AHTTL3MBTL1
SCHEMBL1438626 0.72 RIPK1 (0.41) TSHREPHX2MEN1KMT2AHTT
SCHEMBL5423903 0.72 POLB (0.42) NR1H2S1PR1GLAPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110687-B2 Bicyclic compounds with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-07 US disclosed