SCHEMBL5454293

SCHEMBL5454293

CCOC(=O)CCc1cn(Cc2cc(OCc3ccccc3)cc(OCc3csc(-c4cnccn4)n3)c2)cc1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 4/20 0.37
ALDH1A1 P00352 2/20 0.36
KLKB1 P03952 1/20 0.35
KLK1 P06870 1/20 0.35
PPARG P37231 4/20 0.35
PPARD Q03181 1/20 0.35
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
CPT1B Q92523 1/20 0.34
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
MMP13 P45452 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
TP53 P04637 3/20 0.33
NPC1 O15118 2/20 0.33
NFKB1 P19838 2/20 0.33
RAB9A P51151 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
CDK5 Q00535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5372063 0.97 ALDH1A1 (0.39) PPARAALDH1A1KLKB1KLK1PPARG
SCHEMBL5372440 0.95 F2RL3 (0.38) PPARAALDH1A1KLKB1KLK1PPARG
SCHEMBL5380915 0.95 ALDH1A1 (0.36) PPARAALDH1A1KLKB1KLK1PPARG
SCHEMBL5382597 0.92 ALDH1A1 (0.41) PPARAALDH1A1KLKB1KLK1CPT2
SCHEMBL5384867 0.92 PPARA (0.39) PPARAKLKB1KLK1PPARGCPT2
SCHEMBL5397120 0.90 PPARA (0.38) PPARAALDH1A1KLKB1KLK1PPARG
SCHEMBL5385582 0.89 ALDH1A1 (0.44) PPARAALDH1A1PPARGSMN1; SMN2TP53
SCHEMBL5397102 0.88 ALDH1A1 (0.46) PPARAALDH1A1PPARGSMN1; SMN2TP53
SCHEMBL5377480 0.88 F2RL3 (0.40) PPARAALDH1A1KLKB1KLK1PPARG
SCHEMBL5374473 0.84 ALDH1A1 (0.42) PPARAALDH1A1KLKB1KLK1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179823-B1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-20 US disclosed
EP-1457490-A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity Takeda Chemical Industries, Ltd. (JP) 2004-09-15 EP disclosed
EP-1228067-B1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-07-14 EP disclosed
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed