SCHEMBL545445

SCHEMBL545445

CCCCc1cccc(C(=O)C(OC)C(=O)c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.47
CYP4A11 Q02928 3/20 0.47
PPARA Q07869 4/20 0.47
PPARG P37231 3/20 0.47
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
TRPV1 Q8NER1 1/20 0.41
KAT6A Q92794 1/20 0.41
SPHK2 Q9NRA0 1/20 0.40
SPHK1 Q9NYA1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL633584 0.87 TRPV1 (0.54) TRPV1
SCHEMBL4868007 0.78 PPARA (0.39) PPARACES2CES1
SCHEMBL21887185 0.78 CES2 (0.57) CYP4F2CYP4A11PPARAPPARGCES2
SCHEMBL3387825 0.78 FOLH1 (0.58) CYP4F2CYP4A11PPARAPPARG
SCHEMBL31124111 0.78 FOLH1 (0.58) CYP4F2CYP4A11PPARAPPARG
SCHEMBL28676676 0.77 CYP4F2 (0.57) CYP4F2CYP4A11PPARAPPARGCES2
SCHEMBL146504 0.77 TSHR (0.52) CES2CES1
SCHEMBL30557597 0.77 ELANE (0.40) PPARAPPARG
SCHEMBL1792728 0.77 CYP4A11 (0.75) CYP4F2CYP4A11
SCHEMBL11757933 0.76 CYP4F2 (0.54) CYP4F2CYP4A11PPARAPPARGSPHK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2263788-B1 A PROCESS FOR THE PREPARATION OF MICROCAPSULES FILLED WITH ACTIVE INGREDIENTS SOL GEL TECH LTD (IL) 2018-07-25 EP claimed
EP-1656199-B1 MICROCAPSULES LOADED WITH ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION SOL GEL TECHNOLOGIES LTD (IL) 2016-01-06 EP claimed
US-8110284-B2 Microcapsules loaded with active ingredients and a method for their preparation SOL-GEL TECHNOLOGIES LTD. (IL) 2012-02-07 US claimed
EP-2263788-A2 Microcapsules loaded with active ingredients and a method for their preparation Sol-Gel Technologies Ltd. (IL) 2010-12-22 EP claimed
US-20070292676-A1 Microcapsules Loaded with Active Ingredients and a Method for Their Preparation SOL-GEL TECHNOLOGIES LTD. (IL) 2007-12-20 US claimed
EP-1656199-A1 MICROCAPSULES LOADED WITH ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION Sol-Gel Technologies Ltd. (IL) 2006-05-17 EP claimed
WO-2005009604-A1 MICROCAPSULES LOADED WITH ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION SOL-GEL TECHNOLOGIES LTD. (IL) 2005-02-03 WO claimed
EP-2263788-B1 A PROCESS FOR THE PREPARATION OF MICROCAPSULES FILLED WITH ACTIVE INGREDIENTS SOL GEL TECH LTD (IL) 2018-07-25 EP disclosed
EP-2265243-B1 COOLING COSMETIC OR DERMATOLOGICAL PREPARATIONS HAVING A CONTENT OF (1R,2S,5R)-2-ISOPROPYL-5-METHYL-N-(2-(PYRIDYNE-2-YL)ETHYL-CYCLOHEXANE CARBOXAMIDE AND/OR (1R,2S,5R)-N-(4-(CYANOMETHYL)PHENYL)-2-ISOPROPYL-5- METHYLCYCLOHEXANE CARBOXAMIDE COMPRISING MENTHOXYPROPANE DIOL BEIERSDORF AG (DE) 2017-06-21 EP disclosed
EP-1656199-B1 MICROCAPSULES LOADED WITH ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION SOL GEL TECHNOLOGIES LTD (IL) 2016-01-06 EP disclosed
US-8110284-B2 Microcapsules loaded with active ingredients and a method for their preparation SOL-GEL TECHNOLOGIES LTD. (IL) 2012-02-07 US disclosed
EP-2263788-A2 Microcapsules loaded with active ingredients and a method for their preparation Sol-Gel Technologies Ltd. (IL) 2010-12-22 EP disclosed
US-20100203121-A1 FORMATION OF NANOMETRIC CORE-SHELL PARTICLES HAVING A METAL OXIDE SHELL SOL-GEL TECHNOLOGIES, LTD. (IL) 2010-08-12 US disclosed
EP-2104558-A2 FORMATION OF NANOMETRIC CORE-SHELL PARTICLES HAVING A METAL OXIDE SHELL Sol-Gel Technologies Ltd. (IL) 2009-09-30 EP disclosed
US-20090178692-A1 PERSONAL CLEANSING SYSTEM TAKASAGO INTERNATIONAL CORPORATION (JP) 2009-07-16 US disclosed
EP-2070510-A1 Personal cleansing system Takasago International Corporation (JP) 2009-06-17 EP disclosed
WO-2008072239-A2 FORMATION OF NANOMETRIC CORE-SHELL PARTICLES HAVING A METAL OXIDE SHELL SOL-GEL TECHNOLOGIES LTD. (IL) 2008-06-19 WO disclosed
US-20070292676-A1 Microcapsules Loaded with Active Ingredients and a Method for Their Preparation SOL-GEL TECHNOLOGIES LTD. (IL) 2007-12-20 US disclosed
EP-1656199-A1 MICROCAPSULES LOADED WITH ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION Sol-Gel Technologies Ltd. (IL) 2006-05-17 EP disclosed
WO-2005009604-A1 MICROCAPSULES LOADED WITH ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION SOL-GEL TECHNOLOGIES LTD. (IL) 2005-02-03 WO disclosed