SCHEMBL5466895

SCHEMBL5466895

CCCCC(NS(C)(=O)=O)C(N)c1ccc2c(c1)NC(=O)C(C)O2

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.41
SMYD3 Q9H7B4 4/20 0.38
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.34
MAPK1 P28482 1/20 0.34
MAOB P27338 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5458536 0.80 SMYD3 (0.49) PARP1SMYD3
Hydrochloric Acid SCHEMBL5853934 0.77
SCHEMBL5471771 0.76 SMYD3 (0.42) PARP1SMYD3PDE3BPDE3AMAOB
SCHEMBL5470028 0.75 SMYD3 (0.49) PARP1SMYD3
SCHEMBL6995045 0.74 PARP1 (0.50) PARP1SMYD3PDE3BPDE3AL3MBTL1
SCHEMBL5465453 0.74 SMYD3 (0.50) PARP1SMYD3
SCHEMBL16804878 0.70 PARP1 (0.57) PARP1SMYD3PDE3BPDE3AMAOB
SCHEMBL19966801 0.70 PARP1 (0.57) PARP1SMYD3PDE3BPDE3AMAOB
SCHEMBL5188603 0.68 PARP1 (0.42) PARP1SMYD3PDE3BPDE3AL3MBTL1
SCHEMBL5471775 0.66 SMYD3 (0.42) PARP1SMYD3PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070049583-A1 Benzoxazine and benzothiazine derivatives and their use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 2007-03-01 US disclosed
US-7141566-B1 Benzoxazine and benzothiazine derivatives and the use thereof in medicaments SCHERING AKTIENGESELLSCHAFT (DE) 2006-11-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070049583-A1 Benzoxazine and benzothiazine derivatives and their use in pharmaceutical agents CYP3A5, XDH, CYP4Z1 PARP1 2890/4885SMYD3 4613/4885PDE3B 3180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.