SCHEMBL5481121

SCHEMBL5481121

COC(C)CNC(=O)CN1CCNCC1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.58
CHRM3 P20309 2/20 0.58
SIGMAR1 Q99720 5/20 0.54
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.36
PADI1 Q9ULC6 1/20 0.35
PADI4 Q9UM07 1/20 0.35
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5481706 0.98 CHRM5 (0.56) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL975271 0.80 CHRM5 (0.59) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL1023592 0.75 CHRM5 (0.57) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL4711520 0.75 SIGMAR1 (0.65) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL1904710 0.75 ALDH1A1 (0.69) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL12676423 0.75 CHRM5 (0.53) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL14369164 0.74 SIGMAR1 (0.63) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL10698614 0.74 SIGMAR1 (0.63) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL255190 0.74 CHRM5 (1.00) CHRM5CHRM3SIGMAR1MEN1KMT2A
SCHEMBL2007992 0.73 CHRM5 (0.67) CHRM5CHRM3SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861376-A1 CIS-2,4,5-TRIARYL-IMIDAZOLINES AND THEIR USE AS ANTI-CANCER MEDICAMENTS F. Hoffmann-Roche AG (CH) 2007-12-05 EP disclosed
EP-1753727-A1 NOVEL CIS-IMIDAZOLINES F.HOFFMANN-LA ROCHE AG (CH) 2007-02-21 EP disclosed
WO-2006097261-A1 CIS-2,4,5-TRIARYL-IMIDAZOLINES AND THEIR USE AS ANTI-CANCER MEDICAMENTS F.HOFFMANN-LA ROCHE AG (CH) 2006-09-21 WO disclosed
WO-2005110996-A1 NOVEL CIS-IMIDAZOLINES F.HOFFMANN-LA ROCHE AG (CH) 2005-11-24 WO disclosed