SCHEMBL5481183

SCHEMBL5481183

CC(=O)NCC[Si](C)(C)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.51
MTNR1B P49286 9/20 0.51
MAPT P10636 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CA12 O43570 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ELANE P08246 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6912201 0.79 MAPT (0.55) MTNR1AMTNR1BMAPTL3MBTL1
SCHEMBL5139867 0.78 HDAC3 (0.50) MAPTL3MBTL1CA9
SCHEMBL4395151 0.78 CTSS (0.44) MAPTCA12CA4CA7CA9
SCHEMBL4395154 0.78 CTSS (0.44) MAPTCA12CA4CA7CA9
SCHEMBL9217667 0.75 MAPT (0.47) MAPT
SCHEMBL9243898 0.73 MAPT (0.49) MTNR1AMTNR1BMAPTL3MBTL1HTT
SCHEMBL18238679 0.73 L3MBTL1 (0.51) MTNR1AMTNR1BL3MBTL1
SCHEMBL8719529 0.72 MAPT (0.47) MTNR1AMTNR1BMAPT
SCHEMBL11354893 0.72 MAPT (0.47) MAPTNPSR1
SCHEMBL21294127 0.71 MAPT (0.47) MTNR1AMTNR1BMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737471-A2 PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE OF LIPOPHILIC, SILICON-SUBSTITUTED, CYCLOOXYGENASE-2 SELECTIVE NON-STEROIDAL ANTI-INFLAMMATORY DRUGS AND DERIVATIVES RND Pharmaceuticals (US) 2007-01-03 EP claimed
WO-2005102358-A2 SILICONE-SUBSTITUTED COX-2 SELECTIVE INHIBITORS RND PHARMACEUTICALS (US) 2005-11-03 WO claimed