SCHEMBL5481611

SCHEMBL5481611

FC(F)(F)c1ccc(Nc2cnnc3nc(-c4ncccc4Cl)ccc23)cc1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 18/20 0.59
MAPK3 P27361 1/20 0.47
EPHX2 P34913 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5477967 0.89 TRPV1 (0.76) TRPV1MAPK3
SCHEMBL5477985 0.88 TRPV1 (0.62) TRPV1MAPK3
SCHEMBL5477296 0.86 TRPV1 (0.52) TRPV1MAPK3EPHX2
SCHEMBL5477068 0.84 TRPV1 (0.62) TRPV1MAPK3
SCHEMBL5472596 0.82 TRPV1 (0.66) TRPV1MAPK3
SCHEMBL4678015 0.82 TRPV1 (0.51) TRPV1EPHX2
SCHEMBL5485574 0.80 TRPV1 (0.62) TRPV1EPHX2
SCHEMBL4359111 0.79 TRPV1 (0.54) TRPV1MAPK3EPHX2
SCHEMBL14441331 0.77 TRPV1 (0.59) TRPV1MAPK3
SCHEMBL5479281 0.77 TRPV1 (0.78) TRPV1MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070191374-A1 Substituted cinnolin-4-ylamines NEUROGEN COROPERATION (US) 2007-08-16 US disclosed
US-20070191374-A1 Substituted cinnolin-4-ylamines NEUROGEN COROPERATION (US) 2007-08-16 US disclosed
US-20070191374-A1 Substituted cinnolin-4-ylamines NEUROGEN COROPERATION (US) 2007-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070191374-A1 Substituted cinnolin-4-ylamines CNR1, GPR174, CNR2 TRPV1 379/4885MAPK3 3724/4885EPHX2 2765/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.