SCHEMBL5481861

SCHEMBL5481861

COc1ccc(CO/N=C2\C[C@@H](C(=O)NC[C@@H](O)c3ccccc3)N(C(=O)C(c3ccccc3)c3ccccc3)C2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OXTR P30559 2/20 0.56
AVPR1A P37288 1/20 0.52
AGTR2 P50052 7/20 0.42
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
AGTR1 P30556 2/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP7 P09237 1/20 0.41
MMP13 P45452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4941738 0.90 AGTR2 (0.45) OXTRAGTR2AGTR1MMP1MMP3
SCHEMBL4941744 0.90 AGTR2 (0.45) OXTRAGTR2AGTR1MMP1MMP3
SCHEMBL4942159 0.86 AGTR2 (0.44) OXTRAGTR2AGTR1MMP1MMP3
SCHEMBL4941413 0.85 AGTR2 (0.41) OXTRAGTR2AGTR1MMP1MMP3
SCHEMBL4941411 0.85 AGTR2 (0.41) OXTRAGTR2AGTR1MMP1MMP3
SCHEMBL4944243 0.85 USP2 (0.45) OXTRAGTR2KDM4EGAASMN1; SMN2
SCHEMBL4944248 0.85 USP2 (0.45) OXTRAGTR2KDM4EGAASMN1; SMN2
SCHEMBL4939973 0.81 AGTR2 (0.43) AGTR2GAAAGTR1
SCHEMBL4939969 0.81 AGTR2 (0.43) AGTR2GAAAGTR1
SCHEMBL4941922 0.78 OXTR (0.54) OXTRAVPR1ATDP1MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7211601-B2 Pharmaceutically active pyrrolidine derivatives APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2007-05-01 US claimed