SCHEMBL548191

SCHEMBL548191

COc1cc2c(c(C)c1OC)CC2C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
HTR1A P08908 1/20 0.43
HTR2C P28335 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TPMT P51580 1/20 0.37
ATM Q13315 1/20 0.37
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA9 Q16790 2/20 0.37
CA12 O43570 1/20 0.37
POLB P06746 1/20 0.37
DRD1 P21728 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11215947 0.75 ACHE (0.45) KDM4EALDH1A1HPGDHSD17B10ATM
SCHEMBL547261 0.72 SMN1; SMN2 (0.44) ALDH1A1CA1CA2CA9CA12
SCHEMBL547259 0.72 SMN1; SMN2 (0.44) ALDH1A1CA1CA2CA9CA12
SCHEMBL547260 0.72 SMN1; SMN2 (0.44) ALDH1A1CA1CA2CA9CA12
SCHEMBL31409460 0.72 SMN1; SMN2 (0.44) ALDH1A1CA1CA2CA9CA12
SCHEMBL3034512 0.72 CYP3A4 (0.39) KDM4EALDH1A1HPGDPOLBGAA
SCHEMBL27881140 0.69 KDM4E (0.57) KDM4EALDH1A1HPGDCA1CA2
SCHEMBL9722208 0.67 NQO2 (0.51) KDM4EALDH1A1CA1CA2POLB
SCHEMBL559163 0.67 PARP1 (0.47) KDM4EALDH1A1HPGDCA1CA2
SCHEMBL12586587 0.65 CYP3A4 (0.49) KDM4EALDH1A1HPGDHTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110701-B2 Process for the preparation of functionalised benzocyclobutenes, and application in the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid LES LABORATOIRES SERVIER (FR) 2012-02-07 US disclosed