SCHEMBL5482205

SCHEMBL5482205

C[Si](C)(C)CCCCCCCCC(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOAT1 P35610 2/20 0.43
FAAH O00519 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 2/20 0.39
PAOX Q6QHF9 1/20 0.36
CES2 O00748 3/20 0.33
CES1 P23141 3/20 0.33
TSHR P16473 3/20 0.33
HDAC11 Q96DB2 3/20 0.33
LMNA P02545 1/20 0.33
NFKB1 P19838 1/20 0.33
PMP22 Q01453 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4396869 0.90 SOAT1 (0.37) SOAT1FAAHMEN1KMT2ATP53
SCHEMBL5372245 0.81
SCHEMBL27033087 0.80 TSHR (0.60) MEN1KMT2ATSHRHDAC11LMNA
SCHEMBL7752352 0.80 TSHR (0.60) MEN1KMT2ATSHRHDAC11LMNA
SCHEMBL7595730 0.80 TSHR (0.60) MEN1KMT2ATSHRHDAC11LMNA
SCHEMBL10791260 0.80 TSHR (0.60) MEN1KMT2ATSHRHDAC11LMNA
SCHEMBL9436431 0.80 TSHR (0.60) MEN1KMT2ATSHRHDAC11LMNA
SCHEMBL3960369 0.80 TSHR (0.60) MEN1KMT2ATSHRHDAC11LMNA
SCHEMBL10791818 0.78 TSHR (0.56) FAAHMEN1KMT2ATP53CES2
SCHEMBL25293609 0.78 KMT2A (0.52) SOAT1FAAHMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737471-A2 PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE OF LIPOPHILIC, SILICON-SUBSTITUTED, CYCLOOXYGENASE-2 SELECTIVE NON-STEROIDAL ANTI-INFLAMMATORY DRUGS AND DERIVATIVES RND Pharmaceuticals (US) 2007-01-03 EP claimed
WO-2005102358-A2 SILICONE-SUBSTITUTED COX-2 SELECTIVE INHIBITORS RND PHARMACEUTICALS (US) 2005-11-03 WO claimed