SCHEMBL5484587

SCHEMBL5484587

CCN(CC)CCCC(=O)N1CC(=NOCc2ccc(Cl)c(Cl)c2)C[C@H]1C(=O)NCc1cccc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.37
PEX14 O75381 1/20 0.35
CCR4 P51679 5/20 0.34
MC4R P32245 2/20 0.33
MC1R Q01726 2/20 0.33
MC3R P41968 1/20 0.33
EPHX2 P34913 1/20 0.33
CDYL Q9Y232 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
F2 P00734 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
CYP2C19 P33261 1/20 0.33
CFD P00746 1/20 0.32
MMP1 P03956 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484586 1.00 P2RX7 (0.37) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL5736469 0.93 CCR4 (0.41) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL5736465 0.93 CCR4 (0.41) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL4936450 0.86 P2RX7 (0.40) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL4936458 0.86 P2RX7 (0.40) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL4945653 0.86 P2RX7 (0.42) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL4945655 0.86 P2RX7 (0.42) P2RX7PEX14CCR4MC4RMC1R
SCHEMBL4944148 0.79 GLP1R (0.39) P2RX7PEX14CYP1A2CYP3A4CYP2D6
SCHEMBL4944155 0.79 GLP1R (0.39) P2RX7PEX14CYP1A2CYP3A4CYP2D6
SCHEMBL5743398 0.78 CCR4 (0.41) P2RX7PEX14CCR4EPHX2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7211601-B2 Pharmaceutically active pyrrolidine derivatives APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2007-05-01 US disclosed