SCHEMBL5484715

SCHEMBL5484715

CCc1c[nH]c2cc(N)ccc12.CCc1c[nH]c2cc(N)ccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.51
HTR2C P28335 2/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
IMPDH2 P12268 3/20 0.46
HTR1A P08908 3/20 0.45
HTR1D P28221 2/20 0.45
HTR1B P28222 2/20 0.45
GPR84 Q9NQS5 2/20 0.44
HTR6 P50406 2/20 0.44
CFTR P13569 1/20 0.42
ADRB1 P08588 1/20 0.41
ADRA2A P08913 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR1E P28566 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR7 P34969 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL398434 1.00 HTR2A (0.51) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL3103740 0.85 HPGD (0.62) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL4185239 0.83 HTR2A (0.53) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL5145582 0.83 HTR2A (0.54) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL5742536 0.81 GPR84 (0.49) HTR2AHTR2CMEN1KMT2AHPGD
Dimethylamine SCHEMBL7871287 0.81 HPGD (0.57) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL29507897 0.81 MEN1 (0.60) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL2015074 0.81 HTR2A (0.44) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL27694046 0.81 HTR2A (0.47) HTR2AHTR2CMEN1KMT2AHPGD
SCHEMBL4857335 0.81 MEN1 (0.60) HTR2AHTR2CMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed