SCHEMBL5484987

SCHEMBL5484987

O=C(O)c1c2c(nn1CCCNCCc1ccc(Br)cc1)-c1ccncc1CC2

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.34
CDK2 P24941 4/20 0.33
CCNA2 P20248 3/20 0.33
CCNA1 P78396 3/20 0.33
AURKA O14965 2/20 0.33
NAMPT P43490 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
PDPK1 O15530 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1655852 0.95 AURKA (0.32) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL1656593 0.92 ROCK2 (0.33) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL4270585 0.88 CDK2 (0.33) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL4262255 0.88 ROCK2 (0.38) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL1656607 0.87 CDK2 (0.36) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL4258276 0.87 ROCK2 (0.32) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL4267640 0.87 CCNA2 (0.32) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL4264410 0.87 ROCK2 (0.37) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL4271415 0.87 AURKA (0.32) ROCK2CDK2CCNA2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL1655955 0.87 HTR5A (0.35) ROCK2CDK2CCNA2CCNA1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824498-A2 METHODS AND COMPOSITIONS FOR TREATING CELLULAR PROLIFERATIVE DISEASES THE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2007-08-29 EP disclosed
WO-2006053315-A2 METHODS AND COMPOSITIONS FOR TREATING CELLULAR PROLIFERATIVE DISEASES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2006-05-18 WO disclosed