SCHEMBL5485824

SCHEMBL5485824

CC(=O)Nc1cc([N+](=O)[O-])ccc1Br.CC(=O)OC(C)=O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
CYP19A1 P11511 1/20 0.48
HTT P42858 3/20 0.47
KMT2A Q03164 6/20 0.46
MEN1 O00255 4/20 0.46
CXCR1 P25024 1/20 0.46
CXCR2 P25025 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
GAA P10253 3/20 0.45
EPHX1 P07099 1/20 0.44
PKM P14618 2/20 0.44
CYP1A2 P05177 1/20 0.43
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
DYRK1A Q13627 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL396053 0.93 SMN1; SMN2 (0.57) SMN1; SMN2CYP19A1HTTKMT2AMEN1
SCHEMBL4970698 0.85 SMN1; SMN2 (0.50) SMN1; SMN2CYP19A1HTTKMT2AMEN1
SCHEMBL2311747 0.81 HTT (0.65) SMN1; SMN2HTTKMT2AMEN1CXCR1
SCHEMBL5455180 0.81 GAA (0.64) SMN1; SMN2CYP19A1HTTKMT2AMEN1
SCHEMBL2230525 0.79 KMT2A (0.52) SMN1; SMN2HTTKMT2AMEN1CXCR1
SCHEMBL2230530 0.79 KMT2A (0.52) SMN1; SMN2HTTKMT2AMEN1CXCR1
SCHEMBL30661616 0.79 KMT2A (0.47) SMN1; SMN2HTTKMT2AMEN1CXCR1
SCHEMBL2144447 0.79 KMT2A (0.47) SMN1; SMN2HTTKMT2AMEN1CXCR1
SCHEMBL6318886 0.77 LMNA (0.48) SMN1; SMN2HTTKMT2AMEN1CXCR1
SCHEMBL1008274 0.77 HTT (0.49) SMN1; SMN2HTTKMT2AMEN1CXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed