SCHEMBL5486335

SCHEMBL5486335

CCCc1cccc(C(N)=O)c1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.43
PLA2G2A P14555 6/20 0.42
PLA2G10 O15496 5/20 0.42
HTT P42858 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.40
SLCO1B1 Q9Y6L6 1/20 0.40
LDHA P00338 1/20 0.39
LDHB P07195 1/20 0.39
TSHR P16473 1/20 0.39
HSP90AA1 P07900 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
MEN1 O00255 1/20 0.38
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADRA2A P08913 1/20 0.38
MAPT P10636 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3807642 0.89 BID (0.47) KMT2AMEN1NR1I2LMNACHRM2
SCHEMBL4351825 0.89 BID (0.47) KMT2AMEN1NR1I2LMNACHRM2
SCHEMBL28818542 0.88 TSHR (0.47) HTTLDHALDHBTSHRLTB4R
SCHEMBL28193149 0.86 PLA2G2A (0.49) PLA2G2APLA2G10SIRT2TSHR
SCHEMBL144959 0.84 PARP1 (0.44) KMT2AHTTTSHRMEN1NR1I2
SCHEMBL3352032 0.84 PARP1 (0.41) KMT2AHTTTSHRMEN1NR1I2
Oxalic Acid SCHEMBL27731733 0.83 HMGB1 (0.38) KMT2AHTTMEN1NR1I2LMNA
Oxalic Acid SCHEMBL29264741 0.83 PLA2G2A (0.46) KMT2APLA2G2APLA2G10SIRT2TSHR
Charcoal, Activated SCHEMBL9341326 0.83 PARP1 (0.40) KMT2AHTTTSHRMEN1NR1I2
SCHEMBL6314578 0.83 PARP1 (0.40) KMT2AHTTTSHRMEN1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763509-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2007-03-21 EP disclosed
WO-2006002474-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2006-01-12 WO disclosed